平安! 发表于 2011-11-9 19:57
; e4 P4 `/ U) W! c6 }% yPazopanib (100 mg/kg/day free base equivalent)
8 Q9 y' Z' J' I& H( `+ Y3 { 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。. g# R- x. ~6 U4 F! a6 W d& \
搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。& {& {8 R: ?# A% o% y9 v
! j+ x. t4 O- E. U/ b2 a, m, A e以下是正版说明书的推荐用量。
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--------------------- DOSAGE AND ADMINISTRATION ----------------: I: X5 R% L: \4 L* y" N
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
3 N; F9 z! }, @0 V2 P: E* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) ! ^ q5 a, s h! M0 A4 m/ \
---------------------DOSAGE FORMS AND STRENGTHS --------------
% o! z L* ~" Q, ~200 mg tablets. (3) 8 d3 O- r% X1 y
-------------------------------CONTRAINDICATIONS------------------------ |