平安! 发表于 2011-11-9 19:57
w$ Q; Z9 j& F7 M. c/ uPazopanib (100 mg/kg/day free base equivalent) ; w d' K6 u1 m4 b1 d
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
7 e" f7 n, C# w# G搜索了一下,原料一大堆。1 h, B( i8 x; @0 H% k8 R
! L/ ]2 h, a3 Y6 g' [2 \, o
对不起!100mg/kg是用于移植瘤的,我弄错了。
( D# m: I# a" l+ F5 S# m, ~1 ~8 V, A }9 l$ Z* i( D, Q# A6 Y( B
以下是正版说明书的推荐用量。$ ]% l# y; z: ~" R T: u1 G
: x8 |& @) h4 E--------------------- DOSAGE AND ADMINISTRATION ----------------
) R7 m# I+ N6 H* ^& T+ s: v4 H* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) , L/ D+ x _. u e' ^: M2 Q8 p* E
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 1 Y) s5 j `. d& d( a9 Q) W2 z
---------------------DOSAGE FORMS AND STRENGTHS --------------
4 ^$ O- R* Y/ V7 g200 mg tablets. (3)
8 T* y4 i* W& O9 I7 e/ {-------------------------------CONTRAINDICATIONS------------------------ |